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ARTICLE | Distillery Therapeutics

Therapeutics: P. falciparum plasmepsin I; P. falciparum plasmepsin II; P. falciparum plasmepsin IV

January 7, 2016 8:00 AM UTC

Cell culture studies identified aminoquinazolinone-based inhibitors of Plasmodium falciparum plasmepsins I, II and IV that could help treat malaria. Chemical synthesis and in vitro testing of aminoqui...